Kousuke Hidaka

STING agonist delivery by tumour-penetrating PEG-lipid nanodiscs primes robust anticancer immunity

Eric L. Dane, Alexis Belessiotis‐Richards, Coralie M. Backlund et al. · Nature Materials · 2022 · 320 citations · Full text

Pharmacy, Oncology, Pharmaceutics +17

Discovery of a Novel Series of<i>N</i>-Phenylindoline-5-sulfonamide Derivatives as Potent, Selective, and Orally Bioavailable Acyl CoA:Monoacylglycerol Acyltransferase-2 Inhibitors

Kenjiro Sato, Hiroki Takahagi, Takeshi Yoshikawa et al. · Journal of Medicinal Chemistry · 2015 · 30 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +14

Identification of a novel series of potent and selective CCR6 inhibitors as biological probes

Taisuke Tawaraishi, Nobuki Sakauchi, Kousuke Hidaka et al. · Bioorganic & Medicinal Chemistry Letters · 2018 · 18 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +10

B(OMe)₃ as a Nonacidic Iminium Ion Generator in Mannich‐ and Ugi‐Type Reactions

Yusuke Tanaka, Kousuke Hidaka, Tomoaki Hasui et al. · European Journal of Organic Chemistry · 2009 · 13 citations

Natural Sciences, Chemistry, Catalysis +7

Optimization of a novel series of N-phenylindoline-5-sulfonamide-based acyl CoA:monoacylglycerol acyltransferase-2 inhibitors: Mitigation of CYP3A4 time-dependent inhibition and phototoxic liabilities

Kenjiro Sato, Hiroki Takahagi, Osamu Kubo et al. · Bioorganic & Medicinal Chemistry · 2015 · 11 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +13