Tomoaki Hasui

Identification of Benzoxazin-3-one Derivatives as Novel, Potent, and Selective Nonsteroidal Mineralocorticoid Receptor Antagonists

Tomoaki Hasui, Nobuyuki Matsunaga, Taiichi Ora et al. · Journal of Medicinal Chemistry · 2011 · 109 citations · Full text

Combinatorial Chemistry, Crystal Structure, Medicinal Chemistry +13

Acid-Free, Aminoborane-Mediated Ugi-Type Reaction Leading to General Utilization of Secondary Amines

Yusuke Tanaka, Tomoaki Hasui, Michinori Suginome · Organic Letters · 2007 · 60 citations

Asymmetric Catalysis, General Utilization, Cross-coupling Reaction +14

Synthesis and Reactions of Cyclic Silylboranes

Michinori Suginome, Hiroyoshi Noguchi, Tomoaki Hasui et al. · Bulletin of the Chemical Society of Japan · 2005 · 39 citations

Inorganic Chemistry, Cross-coupling Reaction, Engineering +11

Design, synthesis, and structure–activity relationships of dihydrofuran-2-one and dihydropyrrol-2-one derivatives as novel benzoxazin-3-one-based mineralocorticoid receptor antagonists

Tomoaki Hasui, Taiichi Ohra, Norio Ohyabu et al. · Bioorganic & Medicinal Chemistry · 2013 · 33 citations · Full text

Derivatives, Medicine, Dihydropyrrol-2-one Derivatives +8

Characterization of the binding properties of T-773 as a PET radioligand for phosphodiesterase 10A

Akina Harada, Kazunori Suzuki, Shotaro Miura et al. · Nuclear Medicine and Biology · 2014 · 30 citations

Protein Function, Signal Transduction, Biochemistry +9