Concepedia

Discovery of V-0219: A Small-Molecule Positive Allosteric Modulator of the Glucagon-Like Peptide-1 Receptor toward Oral Treatment for “Diabesity”

Juan Decara, Henar Vázquez‐Villa, José Brea, Mónica Alonso, Raj Kamal Srivastava, Laura Orío, Francisco Alén, Juan Suárez, Elena Baixerás, Javier García‐Cárceles,

Journal of Medicinal Chemistry · 2022 · 21 citations · 13 references

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Abstract

behavior bolsters the interest of a small-molecule PAM of GLP-1R as a promising therapeutic approach for the increasingly prevalent obesity-associated diabetes.

References

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