Concepedia

Design, synthesis and evaluation of covalent inhibitors of DprE1 as antitubercular agents

Lingfeng Liu, Chengcheng Kong, Marco Fumagalli, Karin Savková, Yiwen Xu, Stanislav Huszár, Josè Camilla Sammartino, Dongguang Fan, Laurent R. Chiarelli, Katarı́na Mikus̃ová,

European Journal of Medicinal Chemistry · 2020 · 37 citations · 19 references

DOIFull text

Open access

Concepts

References

19

Bayesian Deconvolution of Mass and Ion Mobility Spectra: From Binary Interactions to Polydisperse Ensembles

Michael T. Marty, Andrew J. Baldwin, Erik G. Marklund et al. · Analytical Chemistry · 2015 · 1.1K citations · Full text

, , +14

Rapid, Low-Technology MIC Determination with Clinical <i>Mycobacterium tuberculosis</i> Isolates by Using the Microplate Alamar Blue Assay

Scott G. Franzblau, Richard Witzig, James C. McLaughlin et al. · Journal of Clinical Microbiology · 1998 · 951 citations · Full text

, , +15

Benzothiazinones Kill <i>Mycobacterium tuberculosis</i> by Blocking Arabinan Synthesis

Vadim Makarov, Giulia Manina, Katarı́na Mikušová et al. · Science · 2009 · 727 citations · Full text

, , +16

Reversible targeting of noncatalytic cysteines with chemically tuned electrophiles

Iana M. Serafimova, Miles A. Pufall, Shyam Krishnan et al. · Nature Chemical Biology · 2012 · 500 citations

, , +12

The discovery of odanacatib (MK-0822), a selective inhibitor of cathepsin K

Jacques Yves Gauthier, Nathalie Chauret, Wanda Cromlish et al. · Bioorganic & Medicinal Chemistry Letters · 2008 · 473 citations · Full text

, , +10