Vadim Makarov

Benzothiazinones Kill <i>Mycobacterium tuberculosis</i> by Blocking Arabinan Synthesis

Vadim Makarov, Giulia Manina, Katarı́na Mikus̃ová et al. · Science · 2009 · 722 citations · Full text

Bioorganic Chemistry, Major Btz Target, Antimicrobial Chemotherapy +18

Towards a new combination therapy for tuberculosis with next generation benzothiazinones

Vadim Makarov, Benoît Lechartier, Ming Zhang et al. · EMBO Molecular Medicine · 2014 · 379 citations · Full text

Pulmonary Tuberculosis, Tuberculosis Prevention, Pharmacology +10

Benzothiazinones: Prodrugs That Covalently Modify the Decaprenylphosphoryl-β-<scp>d</scp>-ribose 2′-epimerase DprE1 of <i>Mycobacterium tuberculosis</i>

Claudia Jessen‐Trefzer, Rengifo-Gonzalez Monica, Marlon J. Hinner et al. · Journal of the American Chemical Society · 2010 · 215 citations · Full text

Bioorganic Chemistry, Antimicrobial Chemotherapy, Chemical Biology +18

Benzothiazinones Are Suicide Inhibitors of Mycobacterial Decaprenylphosphoryl-β-<scp>d</scp>-ribofuranose 2′-Oxidase DprE1

Claudia Jessen‐Trefzer, Henrieta Škovierová, Silvia Buroni et al. · Journal of the American Chemical Society · 2011 · 175 citations · Full text

Bioorganic Chemistry, Btz-resistant Strains, Antimicrobial Chemotherapy +16

Inhibition of Transfer to Secondary Receptors by Heparan Sulfate-Binding Drug or Antibody Induces Noninfectious Uptake of Human Papillomavirus

Hans‐Christoph Selinka, Luise Florin, Hetal D. Patel et al. · Journal of Virology · 2007 · 174 citations · Full text