Design and synthesis of (E)-1,2-diphenylethene-based EZH2 inhibitors

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The polycomb group protein EZH2 is involved in progression of prostate cancer

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EZH2 inhibition as a therapeutic strategy for lymphoma with EZH2-activating mutations

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Medicine, Molecular Genetics, Oncology +15

Durable tumor regression in genetically altered malignant rhabdoid tumors by inhibition of methyltransferase EZH2

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Photochemical preparation of a pyridone containing tetracycle: A jak protein kinase inhibitor

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