Optimization of an azetidine series as inhibitors of colony stimulating factor-1 receptor (CSF-1R) Type II to lead to the clinical candidate JTE-952

Kazutaka Ikegashira, Taku Ikenogami, Takayuki Yamasaki, Takahiro Oka, Yasunori Hase, Naoki Miyagawa, Koji Inagaki, Iichiro Kawahara, Yoshihisa Koga, Hiromasa Hashimoto

Bioorganic & Medicinal Chemistry Letters · 2019 · 14 citations · 13 references

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