Stapled SC34EK fusion inhibitors with high potency against HIV-1 and improved protease resistance

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Life Sciences, Biochemistry, Molecular Biology +14

An All-Hydrocarbon Cross-Linking System for Enhancing the Helicity and Metabolic Stability of Peptides

Christian E. Schafmeister, Julia Po, Gregory L. Verdine · Journal of the American Chemical Society · 2000 · 1K citations

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J Michael Kilby, Sam Hopkins, Thomas M. Venetta et al. · Nature Medicine · 1998 · 994 citations

Life Sciences, Immunology, Molecular Biology +16

Enfuvirtide, an HIV-1 Fusion Inhibitor, for Drug-Resistant HIV Infection in North and South America

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Life Sciences, Pharmacokinetics, Pharmacotherapy +16

Protein Chemical Synthesis by Ligation of Peptide Hydrazides

Ge‐Min Fang, Yi‐Ming Li, Fei Shen et al. · Angewandte Chemie International Edition · 2011 · 798 citations

Life Sciences, Biochemistry, Biocatalysis +7