Concepedia

Metal-free iodine-catalyzed direct cross-dehydrogenative coupling (CDC) between pyrazoles and thiols

Daoshan Yang, Pengfei Sun, Wei Wei, Lingduan Meng, Lingchao He, Baokai Fang, Wei Jiang, Hua Wang

Organic Chemistry Frontiers · 2016 · 58 citations · 68 references

DOI

Concepts

Abstract

A green and efficient iodine-catalyzed cross-dehydrogenative C–S coupling method for the synthesis of C-4 sulfenylated pyrazoles has been initially developed under metal-free conditions.

References

68

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