Concepedia

Novel and potent cyclic cyanamide-based cathepsin K inhibitors

David N. Deaton, Anne M. Hassell, Robert B. McFadyen, Aaron B. Miller, Larry R. Miller, Lisa M. Shewchuk, Francis X. Tavares, Derril H. Willard, Lois L. Wright

Bioorganic & Medicinal Chemistry Letters · 2005 · 42 citations · 13 references

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13

Pycnodysostosis, a Lysosomal Disease Caused by Cathepsin K Deficiency

Bruce D. Gelb, Guo‐Ping Shi, Harold A. Chapman et al. · Science · 1996 · 1K citations

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Collagenase Activity of Cathepsin K Depends on Complex Formation with Chondroitin Sulfate

Zhenqiang Li, Wu-Shiun Hou, Carlos R. Escalante-Torres et al. · Journal of Biological Chemistry · 2002 · 170 citations · Full text

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Potent and Selective Inhibition of Human Cathepsin K Leads to Inhibition of Bone Resorption In Vivo in a Nonhuman Primate

George B. Stroup, Michael W. Lark, Daniel F. Veber et al. · Journal of Bone and Mineral Research · 2001 · 153 citations

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Novel, Nonpeptidic Cyanamides as Potent and Reversible Inhibitors of Human Cathepsins K and L

Jean‐Pierre Falgueyret, Renata M. Oballa, Osamu Okamoto et al. · Journal of Medicinal Chemistry · 2000 · 128 citations · Full text

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Polypeptides. Part XIII. Preparation of α-aza-amino-acid (carbazic acid) derivatives and intermediates for the preparation of α-aza-peptides

Anand S. Dutta, John S. Morley · Journal of the Chemical Society Perkin Transactions 1 · 1975 · 88 citations

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