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Identification of potent type I MetAP inhibitors by simple bioisosteric replacement. Part 1: Synthesis and preliminary SAR studies of thiazole-4-carboxylic acid thiazol-2-ylamide derivatives

Medicinal ChemistryBiochemistryMedicineNatural SciencesPreliminary Sar StudiesRational Drug DesignPharmacotherapyDrug DevelopmentPotent TypePharmacologyPharmaceutical ChemistrySimple Bioisosteric ReplacementDrug Discovery