Concepedia

Development of Homogeneous Nonradioactive Methyltransferase and Demethylase Assays Targeting Histone H3 Lysine 4

Nancy Gauthier, Mireille Caron, Liliana Pedro, Mathieu Arcand, Julie Blouin, Anne Labonté, Claire Normand, Valérie E. Paquet, Anja Rodenbrock, Marjolaine Roy,

SLAS DISCOVERY · 2011 · 41 citations · 28 references

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References

28

A Simple Statistical Parameter for Use in Evaluation and Validation of High Throughput Screening Assays

Ji-Hu Zhang, Thomas D.Y. Chung, Kevin R. Oldenburg · SLAS DISCOVERY · 1999 · 7K citations · Full text

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Histone Demethylation Mediated by the Nuclear Amine Oxidase Homolog LSD1

Yujiang Geno Shi, Yujiang Geno Shi, Fei Lan et al. · Cell · 2004 · 4K citations · Full text

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LSD1 demethylates repressive histone marks to promote androgen-receptor-dependent transcription

Eric Metzger, Melanie Wissmann, Na Yin et al. · Nature · 2005 · 1.7K citations

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MLL Targets SET Domain Methyltransferase Activity to Hox Gene Promoters

Thomas A. Milne, Scott Briggs, Hugh W. Brock et al. · Molecular Cell · 2002 · 1.1K citations · Full text

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Reversal of H3K9me2 by a Small-Molecule Inhibitor for the G9a Histone Methyltransferase

Stefan Kubicek, Roderick J. O’Sullivan, Elias August et al. · Molecular Cell · 2007 · 847 citations

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