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Beta-lactam compounds as apparently uncompetitive inhibitors of HIV-1 protease

Tamás Sperka, J. PITLIK, Péter Bagossi, József Tőzsér

Bioorganic & Medicinal Chemistry Letters · 2005 · 155 citations · 13 references

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13

Comparison of the HIV‐1 and HIV‐2 proteinases using oligopeptide substrates representing cleavage sites in Gag and Gag‐Pol polyproteins

József Tőzsér, Ivo Bláha, Terry D. Copeland et al. · FEBS Letters · 1991 · 161 citations · Full text

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Stability and activity of human immunodeficiency virus protease: comparison of the natural dimer with a homologous, single-chain tethered dimer.

Y S Cheng, F H Yin, S. I. Foundling et al. · Proceedings of the National Academy of Sciences · 1990 · 121 citations

, , +17

The inhibition of human immunodeficiency virus proteases by ‘interface peptides’

Hans J. Schramm, Joachim Boetzel, J. Büttner et al. · Antiviral Research · 1996 · 80 citations

, , +14

The effect of salt on the Michaelis Menten constant of the HIV‐1 protease correlates with the Hofmeister series

Ewald M. Wondrak, John M. Louis, Stephen Oroszlan · FEBS Letters · 1991 · 66 citations · Full text

, , +16

Solid-phase synthesis and SAR of 4-carboxy-2-azetidinone mechanism-based tryptase inhibitors

James Sutton, Scott A. Bolton, Malcolm E. Davis et al. · Bioorganic & Medicinal Chemistry Letters · 2004 · 63 citations · Full text

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