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Introduction of non-natural amino acid residues into the substrate-specific P1 position of trypsin inhibitor SFTI-1 yields potent chymotrypsin and cathepsin G inhibitors

Anna Łęgowska, Dawid Dębowski, Adam Lesner, Magdalena Wysocka, Krzysztof Rolka

Bioorganic & Medicinal Chemistry · 2009 · 44 citations · 24 references

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24

On the size of the active site in proteases. I. Papain

Israël Schechter, Arieh Berger · Biochemical and Biophysical Research Communications · 1967 · 5.2K citations

, , +9

Peptoids: a modular approach to drug discovery.

Reyna J. Simon, Robert S. Kania, Ronald N. Zuckermann et al. · Proceedings of the National Academy of Sciences · 1992 · 941 citations

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p-Nitrophenyl-p′-guanidinobenzoate HCl: A new active site titrant for trypsin

Theodore Chase, Elliott Shaw · Biochemical and Biophysical Research Communications · 1967 · 843 citations

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High-resolution structure of a potent, cyclic proteinase inhibitor from sunflower seeds

S Luckett, R.Santiago Garcia, John J. Barker et al. · Journal of Molecular Biology · 1999 · 398 citations

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Optimization of solid-phase synthesis of [Ala8]-dynorphin A

Nuriá A. Solé, George Bárány · The Journal of Organic Chemistry · 1992 · 208 citations

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