A versatile synthesis of pyrrolo-, furo- and thienopyridines via photocyclization of 3-amino-2-alkene imines in an acid medium

Discovery of a Novel, Potent, and Orally Active Nonpeptide Antagonist of the Human Luteinizing Hormone-Releasing Hormone (LHRH) Receptor

Nobuo Cho, Masataka Harada, Toshihiro Imaeda et al. · Journal of Medicinal Chemistry · 1998 · 126 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +10

The first enantioselective total syntheses of the allopumiliotoxin A alkaloids 267A and 339B

Steven W. Goldstein, Larry E. Overman, Michael H. Rabinowitz · The Journal of Organic Chemistry · 1992 · 83 citations

Pharmacy, Medicinal Chemistry, Pharmacology +7

6-Amino-2-(4-fluorophenyl)-4-methoxy-3- (4-pyridyl)-1<i>H</i>-pyrrolo[2,3-<i>b</i>]pyridine (RWJ 68354):  A Potent and Selective p38 Kinase Inhibitor

James R. Henry, Kenneth C. Rupert, John H. Dodd et al. · Journal of Medicinal Chemistry · 1998 · 77 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +5

A Convenient Method for the Preparation of 5-, 6- and 7-Azaindoles and Their Derivatives

David Hands, Brian Bishop, Mark Cameron et al. · Synthesis · 1996 · 71 citations

Natural Sciences, Chemistry, Medicinal Chemistry +10

Synthesis of tröger's base analogs derived from 3-aminoacridine and 10-aminobenzo[b][1,7]phenanthroline

Hervé Salez, Abderrahim Wardani, Martine Demeunynck et al. · Tetrahedron Letters · 1995 · 45 citations

Pharmacy, Chemistry, Medicinal Chemistry +6