Michael H. Rabinowitz

Enantioselective Total Synthesis of (-)-Ptilomycalin A

Larry E. Overman, Michael H. Rabinowitz, Paul A. Renhowe · Journal of the American Chemical Society · 1995 · 209 citations

Medicinal Chemistry, Molecular Sciences, Chemical Measurement +14

The first enantioselective total syntheses of the allopumiliotoxin A alkaloids 267A and 339B

Steven W. Goldstein, Larry E. Overman, Michael H. Rabinowitz · The Journal of Organic Chemistry · 1992 · 83 citations

Allopumiliotoxin A, Bioorganic Chemistry, Biochemistry +10

Inhibition of tumor necrosis factor-alpha (TNF-alpha) production and arthritis in the rat by GW3333, a dual inhibitor of TNF-alpha-converting enzyme and matrix metalloproteinases.

James G. Conway, Robert Andrews, B Beaudet et al. · PubMed · 2001 · 75 citations

Dual Inhibitor, Soluble Tnf, Tnf-alpha-converting Enzyme +20

Design of Selective and Soluble Inhibitors of Tumor Necrosis Factor-α Converting Enzyme (TACE)

Michael H. Rabinowitz, Robert Andrews, J. David Becherer et al. · Journal of Medicinal Chemistry · 2001 · 73 citations · Full text

Inhibitory Activity, Medicinal Chemistry, Pharmaceutical Science +15

Pharmacological Characterization of 1-(5-Chloro-6-(trifluoromethoxy)-1H-benzoimidazol-2-yl)-1H-pyrazole-4-carboxylic Acid (JNJ-42041935), a Potent and Selective Hypoxia-Inducible Factor Prolyl Hydroxylase Inhibitor

Terrance D. Barrett, Heather L. Palomino, Theresa I. Brondstetter et al. · Molecular Pharmacology · 2011 · 72 citations