Concepedia

Heteroarylaminoethyl and heteroarylthioethyl imidazoles. Synthesis and H3-receptor affinity

Pier Vincenzo Plazzi, Fabrizio Bordi, Marco Mor, Cristiane Sandra da Silva, Giuseppina Morini, Antonio Caretta, Elisabetta Barocelli, T Vitali

European Journal of Medicinal Chemistry · 1995 · 31 citations · 22 references

DOI

Concepts

References

22

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.9K citations

, , +14

Auto-inhibition of brain histamine release mediated by a novel class (H3) of histamine receptor

Jean‐Michel Arrang, M. Garbarg, Jean‐Charles Schwartz · Nature · 1983 · 1.6K citations

, , +14

Highly potent and selective ligands for histamine H3-receptors

J.M. Arrang, M. Garbarg, J.-C. Lancelo et al. · Nature · 1987 · 902 citations

, , +15

Hydrogen Bonding. 33. Factors That Influence the Distribution of Solutes between Blood and Brain

Michael H. Abraham, Harpreet S. Chadha, Robert C. Mitchell · Journal of Pharmaceutical Sciences · 1994 · 301 citations

, , +10

Identification of two H3-histamine receptor subtypes.

Randolph West, Adam Zweig, Neng‐Yang Shih et al. · Molecular Pharmacology · 1990 · 151 citations

, , +16