Auto-inhibition of brain histamine release mediated by a novel class (H3) of histamine receptor

Jean‐Michel Arrang, M. Garbarg, Jean‐Charles Schwartz

Nature

Brain Histamine ReleaseNeurophysiologyMedicineSynaptic TransmissionPhysiology +11

Highly potent and selective ligands for histamine H3-receptors

J.M. Arrang, M. Garbarg, J.-C. Lancelo, +5

Nature

BiochemistryFunctional SelectivityMedicineSelective LigandsReceptor (Biochemistry) +3

Autoinhibition of histamine synthesis mediated by presynaptic H3-receptors

JM Arrang, M. Garbarg, Schwartz Jc

Neuroscience

Molecular PhysiologySignal TransductionBiochemistryMedicineAnesthetic Mechanism +4

Autoregulation of histamine release in brain by presynaptic H3-receptors

J.M. Arrang, M. Garbarg, J.C. Schwartz

Neuroscience

NeurophysiologyNeuropharmacologyNeurologyNeurotransmissionNeuroscience +5

Inhibition of Histamine Synthesis in Brain by α‐Fluoromethylhistidine, a New Irreversible Inhibitor: <i>In Vitro</i> and <i>In Vivo</i> Studies

M. Garbarg, G. Barbin, E. Rodergas, +1

Journal of Neurochemistry

PharmacotherapyExperimental PharmacologyPharmaceutical ChemistrySocial SciencesMolecular Pharmacology +18

Involvement of histaminergic neurons in arousal mechanisms demonstrated with H3-receptor ligands in the cat

Jian‐Sheng Lin, Kazuya Sakai, Giovanna Vanni-Mercier, +4

Brain Research

NeurotransmitterAffective NeuroscienceAnesthetic MechanismNeurotransmissionHistaminergic Neurons +14

A detailed mapping of hist amine H1-receptors in guinea-pig central nervous system established by autoradiography with [125I]iodobolpyramine

Marie-Louise Bouthenet, Martial Ruat, N. Salès, +2

Neuroscience

Hist Amine H1-receptorsNeurophysiologyNeuroanatomyMedicineNeuropeptide Receptor +9

Histaminergic Pathway in Rat Brain Evidenced by Lesions of the Medial Forebrain Bundle

M. Garbarg, G. Barbin, Jean Féger, +1

Science

Histaminergic PathwayMedial Forebrain BundleNeurophysiologyNeuroanatomyPhysiology +12

Actions of betahistine at histamine receptors in the brain

Jean‐Michel Arrang, M. Garbarg, Tam Thanh Quach, +3

European Journal of Pharmacology

NeurophysiologyMedicineNeurotransmitterNeuropharmacologyNeuroscience +6

S-[2-(4-imidazolyl)ethyl]isothiourea, a highly specific and potent histamine H3 receptor agonist.

M. Garbarg, J.M. Arrang, A. Rouleau, +4

Journal of Pharmacology and Experimental Therapeutics