Bioorganic & Medicinal Chemistry Letters · 1998 · 42 citations · 25 references
MedicineMedicinal ChemistryPharmacologyDrug DesignEnzymologyMolecular PharmacologyCardiac MedicationsConformational SamplingDrug-receptor InteractionsEnzyme InhibitionEnzyme-substrate RecognitionLigand BindingCaptopril TherapyConformational EquilibriumConformational MappingEnzyme ActivityEnzyme Activity RegulationRenin-angiotensin System ModulationRenin-angiotensin-aldosterone System Inhibition
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A new class of angiotensin-converting enzyme inhibitors
Arthur A. Patchett, Elbert E. Harris, Edward W. Tristram et al. · Nature · 1980 · 706 citations