Design, synthesis, and evaluation of 5-methyl-4-phenoxy-5H-pyrrolo[3,2-d]pyrimidine derivatives: Novel VEGFR2 kinase inhibitors binding to inactive kinase conformation

Yuya Oguro, Naoki Miyamoto, Kengo Okada, Terufumi Takagi, Hidehisa Iwata, Yoshiko Awazu, Hiroshi Miki, Akira Hori, Keiji Kamiyama, Shinichi Imamura

Bioorganic & Medicinal Chemistry · 2010 · 122 citations · 16 references

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