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Subtype-selective Nav1.8 sodium channel blockers: Identification of potent, orally active nicotinamide derivatives

Michael E. Kort, Robert N. Atkinson, James B. Thomas, Irene Drizin, Matthew S. Johnson, Matthew A. Secrest, Robert J. Gregg, Marc J. C. Scanio, Lei Shi, Ahmed H. Hakeem,

Bioorganic & Medicinal Chemistry Letters · 2010 · 28 citations · 10 references

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An experimental model for peripheral neuropathy produced by segmental spinal nerve ligation in the rat

Sun Ho Kim, Jin Mo Chung · Pain · 1992 · 3K citations

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Palladium‐Catalyzed Cross‐Coupling Reactions in Total Synthesis

K. C. Nicolaou, Paul G. Bulger, David Šarlah · Angewandte Chemie International Edition · 2005 · 2.7K citations

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A-803467, a potent and selective Na <sub>v</sub> 1.8 sodium channel blocker, attenuates neuropathic and inflammatory pain in the rat

Michael F. Jarvis, Prisca Honoré, Char‐Chang Shieh et al. · Proceedings of the National Academy of Sciences · 2007 · 514 citations · Full text

Cross‐Coupling Reactions on Azoles with Two and More Heteroatoms

Michael Schnürch, Radoslav Flašík, Ather Farooq Khan et al. · European Journal of Organic Chemistry · 2006 · 279 citations

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Discovery, Synthesis, and Bioactivity of Bis(heteroaryl)piperazines. 1. A Novel Class of Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitors

Donna L. Romero, Raymond A. Morge, Carolyn Biles et al. · Journal of Medicinal Chemistry · 1994 · 90 citations

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