Concepedia

A regiospecific synthesis of a series of 1-sulfonyl azepinoindoles as potent 5-HT6 ligands

Kevin G. Liu, Jennifer R. Lo, Thomas A. Comery, Guo Ming Zhang, Jean Y. Zhang, Dianne Kowal, Deborah L. Smith, Li Di, Edward H. Kerns, Lee E. Schechter,

Bioorganic & Medicinal Chemistry Letters · 2008 · 26 citations · 6 references

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6

Discovery of 5-Arylsulfonamido-3- (pyrrolidin-2-ylmethyl)-1<i>H</i>-indole Derivatives as Potent, Selective 5-HT<sub>6</sub>Receptor Agonists and Antagonists

Derek C. Cole, William J. Lennox, Sabrina Lombardi et al. · Journal of Medicinal Chemistry · 2004 · 102 citations · Full text

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N1-(Benzenesulfonyl)tryptamines as novel 5-HT6 antagonists

Yuching Tsai, Maƚgorzata Dukat, Abdelmalik Slassi et al. · Bioorganic & Medicinal Chemistry Letters · 2000 · 92 citations · Full text

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<i>N</i>-Arylsulfonylindole Derivatives as Serotonin 5-HT<sub>6</sub>Receptor Ligands

Michael G. N. Russell, Robert J. Baker, Laura M. Barden et al. · Journal of Medicinal Chemistry · 2001 · 92 citations · Full text

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Rearrangement of 3,3-Disubstituted Indolenines and Synthesis of 2,3-Substituted Indoles

Kevin G. Liu, Albert J. Robichaud, Jennifer R. Lo et al. · Organic Letters · 2006 · 77 citations · Full text

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N1-arylsulfonyl-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole derivatives are potent and selective 5-HT6 receptor antagonists

Derek C. Cole, John W. Ellingboe, William J. Lennox et al. · Bioorganic & Medicinal Chemistry Letters · 2004 · 43 citations · Full text

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