Michael G. N. Russell

Fluorination of 3-(3-(Piperidin-1-yl)propyl)indoles and 3-(3-(Piperazin-1-yl)propyl)indoles Gives Selective Human 5-HT_1D Receptor Ligands with Improved Pharmacokinetic Profiles

Monique B. van Niel, Ian Collins, Margaret S. Beer et al. · Journal of Medicinal Chemistry · 1999 · 157 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +16

<i>N</i>-Arylsulfonylindole Derivatives as Serotonin 5-HT₆Receptor Ligands

Michael G. N. Russell, Robert J. Baker, Laura M. Barden et al. · Journal of Medicinal Chemistry · 2001 · 92 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +17

Controlled Modification of Acidity in Cholecystokinin B Receptor Antagonists:  <i>N</i>-(1,4-Benzodiazepin-3-yl)-<i>N</i> ‘-[3-(tetrazol-5-ylamino)phenyl]ureas

José L. Castro, Richard G. Ball, Howard B. Broughton et al. · Journal of Medicinal Chemistry · 1996 · 69 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +16

Discovery of Functionally Selective 7,8,9,10-Tetrahydro-7,10-ethano-1,2,4-triazolo[3,4-<i>a</i>]phthalazines as GABA_AReceptor Agonists at the α₃Subunit

Michael G. N. Russell, Robert W. Carling, John Atack et al. · Journal of Medicinal Chemistry · 2005 · 61 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +17

Synthesis and Biological Activity of 3-[2-(Dimethylamino)ethyl]-5-[(1,1-dioxo-5-methyl-1,2,5-thiadiazolidin-2-yl)methyl]-1H-indole and Analogs: Agonists for the 5-HT1D Receptor

José L. Castro, Raymond Baker, Alexander R. Guiblin et al. · Journal of Medicinal Chemistry · 1994 · 61 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +10