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An investigation into the structure–activity relationships associated with the systematic modification of the β2-adrenoceptor agonist indacaterol

David T. Beattie, David Beer, Michelle Bradley, Ian C. Bruce, Steven J. Charlton, Bernard Cuenoud, Robin A. Fairhurst, David Farr, John R. Fozard, Diana Janus,

Bioorganic & Medicinal Chemistry Letters · 2012 · 34 citations · 19 references

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References

19

Crystal structure of the human β2 adrenergic G-protein-coupled receptor

Søren G. F. Rasmussen, Hee‐Jung Choi, Daniel M. Rosenbaum et al. · Nature · 2007 · 1.9K citations

, , +16

Structure of a nanobody-stabilized active state of the β2 adrenoceptor

Søren G. F. Rasmussen, Hee‐Jung Choi, Juan José Fung et al. · Nature · 2011 · 1.7K citations · Full text

, , +6

Cloning of the gene and cDNA for mammalian β-adrenergic receptor and homology with rhodopsin

Richard A. F. Dixon, Brian K. Kobilka, David J. Strader et al. · Nature · 1986 · 1.3K citations

, , +8

Sequential Binding of Agonists to the β2 Adrenoceptor

Gayathri Swaminath, Yang K. Xiang, Tae Weon Lee et al. · Journal of Biological Chemistry · 2003 · 331 citations · Full text

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Involvement of Asn-293 in stereospecific agonist recognition and in activation of the beta 2-adrenergic receptor.

Kerstin Wieland, H. M. ZUURMOND, Cornelius Krasel et al. · Proceedings of the National Academy of Sciences · 1996 · 196 citations

, , +17