Concepedia

In vitro plasma stability, permeability and solubility of mercaptoacetamide histone deacetylase inhibitors

Roula Konsoula, Mira Jung

International Journal of Pharmaceutics · 2008 · 105 citations · 29 references

DOI

Concepts

References

29

A Theoretical Basis for a Biopharmaceutic Drug Classification: The Correlation of in Vitro Drug Product Dissolution and in Vivo Bioavailability

Gordon L. Amidon, Hans Lennernäs, Vinod P. Shah et al. · Pharmaceutical Research · 1995 · 5.3K citations · Full text

, , +16

Correlation between oral drug absorption in humans and apparent drug permeability coefficients in human intestinal epithelial (Caco-2) cells

Per Artursson, Johan Karlsson · Biochemical and Biophysical Research Communications · 1991 · 1.9K citations

, , +16

Phase I Study of an Oral Histone Deacetylase Inhibitor, Suberoylanilide Hydroxamic Acid, in Patients With Advanced Cancer

William Kevin Kelly, Owen A. O’Connor, Lee M. Krug et al. · Journal of Clinical Oncology · 2005 · 907 citations · Full text

, , +16

Molecular Properties of WHO Essential Drugs and Provisional Biopharmaceutical Classification

Nehal A. Kasim, Marc Whitehouse, Chandrasekharan Ramachandran et al. · Molecular Pharmaceutics · 2003 · 844 citations

, , +16

FK228 (depsipeptide) as a natural prodrug that inhibits class I histone deacetylases.

Ryohei Furumai, Akihisa Matsuyama, Nobuyuki Kobashi et al. · PubMed · 2002 · 744 citations

, , +13