Concepedia

Identification and optimization of a novel series of [2.2.1]-oxabicyclo imide-based androgen receptor antagonists

Mark Salvati, Aaron Balog, Weifang Shan, Richard Rampulla, Sören Giese, Tom Mitt, Joseph A. Furch, Gregory D. Vite, Ricardo M. Attar, Maria Jure–Kunkel,

Bioorganic & Medicinal Chemistry Letters · 2008 · 34 citations · 16 references

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16

Cancer Statistics, 2002

Ahmedin Jemal, Anish Thomas, Thomas S. Murray et al. · CA A Cancer Journal for Clinicians · 2002 · 2.9K citations · Full text

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Molecular determinants of resistance to antiandrogen therapy

Charlie D. Chen, Derek S. Welsbie, Chris Tran et al. · Nature Medicine · 2003 · 2.3K citations

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STUDIES ON PROSTATIC CANCER

Charles Huggins · Archives of surgery · 1941 · 1.5K citations

, , +10

Crystallographic structures of the ligand-binding domains of the androgen receptor and its T877A mutant complexed with the natural agonist dihydrotestosterone

John S. Sack, Kevin Kish, Chihuei Wang et al. · Proceedings of the National Academy of Sciences · 2001 · 485 citations · Full text

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Flexible protein–ligand docking by global energy optimization in internal coordinates

Maxim Totrov, Ruben Abagyan · Proteins Structure Function and Bioinformatics · 1997 · 408 citations

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