Kevin Kish

The Structure of Dasatinib (BMS-354825) Bound to Activated ABL Kinase Domain Elucidates Its Inhibitory Activity against Imatinib-Resistant ABL Mutants

John S. Tokarski, John A. Newitt, Chieh Ying J. Chang et al. · Cancer Research · 2006 · 686 citations · Full text

Medicine, Medicinal Chemistry, Oncology +13

Crystallographic structures of the ligand-binding domains of the androgen receptor and its T877A mutant complexed with the natural agonist dihydrotestosterone

John S. Sack, Kevin Kish, Chihuei Wang et al. · Proceedings of the National Academy of Sciences · 2001 · 485 citations · Full text

Life Sciences, Biochemistry, Endocrinology +17

Potent and selective biphenyl azole inhibitors of adipocyte fatty acid binding protein (aFABP)

Richard Sulsky, David R. Magnin, Yanting Huang et al. · Bioorganic & Medicinal Chemistry Letters · 2006 · 151 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +13

Pharmacological and X-Ray Structural Characterization of a Novel Selective Androgen Receptor Modulator: Potent Hyperanabolic Stimulation of Skeletal Muscle with Hypostimulation of Prostate in Rats

Jacek Ostrowski, Joyce E. Kuhns, John A. Lupisella et al. · Endocrinology · 2006 · 129 citations

Medicine, Endocrinology, Pharmacology +17

Involvement of DPP‐IV catalytic residues in enzyme–saxagliptin complex formation

William J. Metzler, Joseph Yanchunas, Carolyn A. Weigelt et al. · Protein Science · 2008 · 128 citations · Full text

Life Sciences, Biochemistry, Pharmacology +17