Design and synthesis of N-methylpyrimidone derivatives as HIV-1 integrase inhibitors

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Life Sciences, Genetics, Molecular Biology +16

Requirement for Integrase during Reverse Transcription of Human Immunodeficiency Virus Type 1 and the Effect of Cysteine Mutations of Integrase on Its Interactions with Reverse Transcriptase

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Life Sciences, Genetics, Molecular Biology +14

The use of oxadiazole and triazole substituted naphthyridines as HIV-1 integrase inhibitors. Part 1: Establishing the pharmacophore

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