Intrinsic Absolute Bioavailability Prediction in Rats Based on In Situ Absorption Rate Constants and/or In Vitro Partition Coefficients: 6‐Fluoroquinolones

A Theoretical Basis for a Biopharmaceutic Drug Classification: The Correlation of in Vitro Drug Product Dissolution and in Vivo Bioavailability

Gordon L. Amidon, Hans Lennernäs, Vinod P. Shah et al. · Pharmaceutical Research · 1995 · 5.3K citations · Full text

Pharmacy, Pharmacokinetics, Pharmacology +16

Some suggestions for measuring predictive performance

Lewis B. Sheiner, Stuart L. Beal · Journal of Pharmacokinetics and Biopharmaceutics · 1981 · 1.6K citations

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Drug Absorption I: An In Situ Rat Gut Technique Yielding Realistic Absorption Rates

James T. Doluisio, Norman F. Billups, Lewis W. Dittert et al. · Journal of Pharmaceutical Sciences · 1969 · 349 citations

Pharmacy, Pharmacokinetics, Pharmacology +12

Predicting Fraction Dose Absorbed in Humans Using a Macroscopic Mass Balance Approach

Patrick J. Sinko, Glen Leesman, Gordon L. Amidon · Pharmaceutical Research · 1991 · 176 citations · Full text

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Studies on the reliability of a bihyperbolic functional absorption model. I. Ring-substituted anilines

A. Martín‐Villodre, J.M. Plá-Delfina, Joaquín Moreno et al. · Journal of Pharmacokinetics and Biopharmaceutics · 1986 · 74 citations

Natural Sciences, Chemistry, Physics +6