(4-Phenoxyphenyl)tetrazolecarboxamides and related compounds as dual inhibitors of fatty acid amide hydrolase (FAAH) and monoacylglycerol lipase (MAGL)

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Modulation of anxiety through blockade of anandamide hydrolysis

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Selective blockade of 2-arachidonoylglycerol hydrolysis produces cannabinoid behavioral effects

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Discovering potent and selective reversible inhibitors of enzymes in complex proteomes

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Life Sciences, Biochemistry, Medicinal Chemistry +11

Characterization of Monoacylglycerol Lipase Inhibition Reveals Differences in Central and Peripheral Endocannabinoid Metabolism

Jonathan Z. Long, Daniel K. Nomura, Benjamin F. Cravatt · Chemistry & Biology · 2009 · 310 citations · Full text

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