Concepedia

The development and SAR of pyrrolidine carboxamide 11β-HSD1 inhibitors

Hengmiao Cheng, Jacqui Hoffman, Phuong Le, Sajiv K. Nair, Stephan J. Cripps, Jean Matthews, Christopher Smith, Michele Yang, Stan Kupchinsky, Klaus Dress,

Bioorganic & Medicinal Chemistry Letters · 2010 · 44 citations · 16 references

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16

A Transgenic Model of Visceral Obesity and the Metabolic Syndrome

Hiroaki Masuzaki, J. Paterson, Hiroshi Shinyama et al. · Science · 2001 · 1.8K citations

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Mineralocorticoid Action: Target Tissue Specificity Is Enzyme, Not Receptor, Mediated

John W. Funder, P. Pearce, A. Ian Smith · Science · 1988 · 1.6K citations

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LOCALISATION OF 11β-HYDROXYSTEROID DEHYDROGENASE—TISSUE SPECIFIC PROTECTOR OF THE MINERALOCORTICOID RECEPTOR

Christopher R.W. Edwards, D. Burt, Martin McIntyre et al. · The Lancet · 1988 · 1.1K citations · Full text

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11β-Hydroxysteroid dehydrogenase type 1 knockout mice show attenuated glucocorticoid-inducible responses and resist hyperglycemia on obesity or stress

Yuri Kotelevtsev, Megan C. Holmes, Ann N. Burchell et al. · Proceedings of the National Academy of Sciences · 1997 · 855 citations

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Purification and Characterization of the Corticosteroid 1lβ-Dehydrogenase Component of the Rat Liver 1lβ-Hydroxysteroid Dehydrogenase Complex*

Vijaya M. Lakshmi, Carl Monder · Endocrinology · 1988 · 311 citations

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