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Antagonists of the human adenosine A2A receptor. Part 2: Design and synthesis of 4-arylthieno[3,2-d]pyrimidine derivatives

Roger J. Gillespie, Ian A. Cliffe, Claire Dawson, Colin T. Dourish, Suneel Gaur, Paul R. Giles, Allan M. Jordan, Antony R. Knight, Anthony J. Lawrence, Joanne Lerpiniere,

Bioorganic & Medicinal Chemistry Letters · 2008 · 32 citations · 6 references

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Functional characterization of agonists at recombinant human 5‐HT<sub>2A</sub>, 5‐HT<sub>2B</sub> and 5‐HT<sub>2C</sub> receptors in CHO‐K1 cells

Richard H. Porter, Karen Benwell, Helen Lamb et al. · British Journal of Pharmacology · 1999 · 356 citations · Full text

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Discovery of nonxanthine adenosine A<sub>2A</sub>receptor antagonists for the treatment of Parkinson’s disease

Scott Μ. Weiss, Karen Benwell, Ian A. Cliffe et al. · Neurology · 2003 · 77 citations

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Antagonists of the human adenosine A2A receptor. Part 3: Design and synthesis of pyrazolo[3,4-d]pyrimidines, pyrrolo[2,3-d]pyrimidines and 6-arylpurines

Roger J. Gillespie, Ian A. Cliffe, Claire Dawson et al. · Bioorganic & Medicinal Chemistry Letters · 2008 · 65 citations · Full text

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Adenosine A2 receptors modulate haloperidol-induced catalepsy in rats

Sanjay N. Mandhane, Chandrabhan T. Chopde, Anuradha K Ghosh · European Journal of Pharmacology · 1997 · 60 citations

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Antagonists of the human adenosine A2A receptor. Part 1: Discovery and synthesis of thieno[3,2-d]pyrimidine-4-methanone derivatives

Roger J. Gillespie, David R. Adams, David Bebbington et al. · Bioorganic & Medicinal Chemistry Letters · 2008 · 48 citations · Full text

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