[³H]MK‐801 Labels a Site on the <i>N</i>‐Methyl‐D‐Aspartate Receptor Channel Complex in Rat Brain Membranes

Erik H.F. Wong, Antony R. Knight, Geoffrey N. Woodruff

Journal of Neurochemistry

Antagonists of the human adenosine A2A receptor. Part 3: Design and synthesis of pyrazolo[3,4-d]pyrimidines, pyrrolo[2,3-d]pyrimidines and 6-arylpurines

Roger J. Gillespie, Ian A. Cliffe, Claire Dawson, +12

Bioorganic & Medicinal Chemistry Letters

BiochemistryMedicineMechanism Of ActionReceptor (Biochemistry)Pharmacological Agent +3

Antagonists of the human adenosine A2A receptor. Part 1: Discovery and synthesis of thieno[3,2-d]pyrimidine-4-methanone derivatives

Roger J. Gillespie, David R. Adams, David Bebbington, +20

Bioorganic & Medicinal Chemistry Letters

Molecular PharmacologyBiochemistryFunctional SelectivityMedicineReceptor (Biochemistry) +4

Antagonists of the human adenosine A2A receptor. Part 2: Design and synthesis of 4-arylthieno[3,2-d]pyrimidine derivatives

Roger J. Gillespie, Ian A. Cliffe, Claire Dawson, +13

Bioorganic & Medicinal Chemistry Letters

Molecular PharmacologyBiochemistryMedicineMechanism Of ActionReceptor (Biochemistry) +4

Pyrrolo(iso)quinoline derivatives as 5-HT2C receptor agonists

David R. Adams, Jonathan Bentley, Karen Benwell, +13

Bioorganic & Medicinal Chemistry Letters

Molecular PharmacologyBiochemistryFunctional SelectivityMedicineReceptor (Biochemistry) +5

Characterisation of agonist binding on human 5-HT2C receptor isoforms

Kathleen Quirk, Anthony J. Lawrence, J. Alison Jones, +6

European Journal of Pharmacology

Molecular PharmacologySignal TransductionG Protein-coupled ReceptorMedicineFunctional Selectivity +5

Identification of non-furan containing A2A antagonists using database mining and molecular similarity approaches

Christine M. Richardson, Roger J. Gillespie, D.S. Williamson, +5

Bioorganic & Medicinal Chemistry Letters

Medicinal ChemistryDatabase MiningDrug TargetBiochemistryMedicine +10

Discovery and functional evaluation of diverse novel human CB1 receptor ligands

Nicolas Foloppe, Karen Benwell, Teresa Brooks, +4

Bioorganic & Medicinal Chemistry Letters

Cannabis UseFunctional EvaluationDrug TargetFunctional SelectivityMedicine +5

5-HT2C Receptor Agonists for the Treatment of Obesity. Biological and Chemical Adventures

David Adams, Sven Taylor, Stephan Röver, +14

CHIMIA International Journal for Chemistry

Food IntakePeptide ScienceChemical BiologyPharmaceutical ChemistryPyrroloindole Core +23

Discovery of a novel class of selective human CB1 inverse agonists

Nicolas Foloppe, Nicola H. Allen, Carol H. Bentley, +7

Bioorganic & Medicinal Chemistry Letters

Cannabis UseDrug TargetFunctional SelectivityMedicineReceptor (Biochemistry) +7