Roger J. Gillespie

Antagonists of the Human A_2A Adenosine Receptor. 4. Design, Synthesis, and Preclinical Evaluation of 7-Aryltriazolo[4,5-<i>d</i>]pyrimidines

Roger J. Gillespie, Samantha J. Bamford, Ruth Botting et al. · Journal of Medicinal Chemistry · 2008 · 103 citations · Full text

Medicine, Pharmacokinetics, Pharmacology +15

Antagonists of the human adenosine A2A receptor. Part 3: Design and synthesis of pyrazolo[3,4-d]pyrimidines, pyrrolo[2,3-d]pyrimidines and 6-arylpurines

Roger J. Gillespie, Ian A. Cliffe, Claire Dawson et al. · Bioorganic & Medicinal Chemistry Letters · 2008 · 65 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +12

A novel application of the Dess-Martin reagent to the synthesis of an FK506 analogue and other tricarbonyl compounds

Mark Batchelor, Roger J. Gillespie, Julian M.C. Golec et al. · Tetrahedron Letters · 1993 · 63 citations

Natural Sciences, Chemistry, Medicinal Chemistry +8

Rhodium(II)-catalysed addition of dimethyl diazomalonate to thiophen: a simple synthesis of thiophenium bismethoxycarbonylmethylides and crystal and molecular structure of the unsubstituted methylide

Roger J. Gillespie, Judith Murray‐Rust, Peter Murray‐Rust et al. · Journal of the Chemical Society Chemical Communications · 1978 · 52 citations

Natural Sciences, Biochemistry, Chemistry +13

Antagonists of the human adenosine A2A receptor. Part 1: Discovery and synthesis of thieno[3,2-d]pyrimidine-4-methanone derivatives

Roger J. Gillespie, David R. Adams, David Bebbington et al. · Bioorganic & Medicinal Chemistry Letters · 2008 · 48 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +11