Suneel Gaur

Antagonists of the Human A_2A Adenosine Receptor. 4. Design, Synthesis, and Preclinical Evaluation of 7-Aryltriazolo[4,5-<i>d</i>]pyrimidines

Roger J. Gillespie, Samantha J. Bamford, Ruth Botting et al. · Journal of Medicinal Chemistry · 2008 · 103 citations · Full text

Molecular Pharmacology, Medicinal Chemistry, Striatal Dopamine +14

Antagonists of the human adenosine A2A receptor. Part 3: Design and synthesis of pyrazolo[3,4-d]pyrimidines, pyrrolo[2,3-d]pyrimidines and 6-arylpurines

Roger J. Gillespie, Ian A. Cliffe, Claire Dawson et al. · Bioorganic & Medicinal Chemistry Letters · 2008 · 65 citations · Full text

Biochemistry, Medicine, Mechanism Of Action +5

Enantiospecific preparation of [(2r,6s)-endo]-5-aza-1,10,10-trimethyl-3-oxatricyclo[5.2.1.02,6]decan-4-one by a nitrene-mediated route from [(1s)-endo]-(−)-borneol and its utility as a chiral auxiliary in some asymmetric transformations

Malcolm R. Banks, Alexander J. Blake, J. I. G. Cadogan et al. · Tetrahedron · 1992 · 51 citations

Enantioselective Synthesis, Engineering, Natural Sciences +9

Antagonists of the human adenosine A2A receptor. Part 1: Discovery and synthesis of thieno[3,2-d]pyrimidine-4-methanone derivatives

Roger J. Gillespie, David R. Adams, David Bebbington et al. · Bioorganic & Medicinal Chemistry Letters · 2008 · 48 citations · Full text

Molecular Pharmacology, Biochemistry, Functional Selectivity +6

Indoline derivatives as 5-HT 2C receptor agonists

Jonathan Bentley, David R. Adams, David Bebbington et al. · Bioorganic & Medicinal Chemistry Letters · 2004 · 44 citations · Full text

Functional Selectivity, Medicine, Physiology +5