Concepedia

Discovery of FR166124, a novel water-soluble pyrazolo-[1,5-α]pyridine adenosine A1 receptor antagonist

Satoru Kuroda, Atsushi Akahane, Hiromichi Itani, Shintaro Nishimura, Kieran Durkin, Takayoshi Kinoshita, Yoshiyuki Tenda, Kazuo Sakane

Bioorganic & Medicinal Chemistry Letters · 1999 · 44 citations · 9 references

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9

Binding of the A1-selective adenosine antagonist 8-cyclopentyl-1,3-dipropylxanthine to rat brain membranes

Robert F. Bruns, James H. Fergus, Edward W. Badger et al. · Naunyn-Schmiedeberg s Archives of Pharmacology · 1987 · 377 citations

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Adenosine Receptor Antagonists: Structures and Potential Therapeutic Applications

Christa E. Müller, Birgitt Stein · Current Pharmaceutical Design · 1996 · 123 citations

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Discovery of 6-Oxo-3-(2-phenylpyrazolo[1,5-<i>a</i>]pyridin-3-yl)-1(6<i>H</i>)-pyridazinebutanoic Acid (FK 838):  A Novel Non-Xanthine Adenosine A<sub>1</sub>Receptor Antagonist with Potent Diuretic Activity

Atsushi Akahane, Hirohito Katayama, Takafumi Mitsunaga et al. · Journal of Medicinal Chemistry · 1999 · 102 citations · Full text

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Solubilities of Adenosine Antagonists Determined by Radioreceptor Assay

Robert F. Bruns, James H. Fergus · Journal of Pharmacy and Pharmacology · 1989 · 41 citations

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Discovery of FK453, a novel non-xanthine adenosine A1 receptor antagonist

Atsushi Akahane, Hirohito Katayama, Takafumi Mitsunaga et al. · Bioorganic & Medicinal Chemistry Letters · 1996 · 28 citations

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