Kieran Durkin

Antineoplastic agents 337. Synthesis of dolastatin 10 structural modifications.

George R. Pettit, Jayaram K. Srirangam, József Barkóczy et al. · PubMed · 1995 · 70 citations

Medicine, Oncology, Pharmacology +17

Discovery of FR166124, a novel water-soluble pyrazolo-[1,5-α]pyridine adenosine A1 receptor antagonist

Satoru Kuroda, Atsushi Akahane, Hiromichi Itani et al. · Bioorganic & Medicinal Chemistry Letters · 1999 · 44 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +10

3-Amino-pyrazolo[3,4-d]pyrimidines as p38α kinase inhibitors: Design and development to a highly selective lead

Michael Soth, Sarah C. Abbot, Allassan Abubakari et al. · Bioorganic & Medicinal Chemistry Letters · 2011 · 27 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +14

Novel adenosine A1 receptor antagonists. Synthesis and structure–activity relationships of a novel series of 3-(2-cyclohexenyl-3-oxo-2,3-dihydropyridazin-6-yl)-2-phenylpyrazolo[1,5-a]pyridines

Satoru Kuroda, Atsushi Akahane, Hiromichi Itani et al. · Bioorganic & Medicinal Chemistry · 2000 · 20 citations

Medicine, Medicinal Chemistry, Pharmacology +16

Synthesis of the water-soluble adenosine A1 receptor antagonist FR166124 through a novel sequential Horner-Emmons / isomerization reaction

Satoru Kuroda, Atsushi Akahane, Hiromichi Itani et al. · Tetrahedron · 1999 · 10 citations

Medicine, Medicinal Chemistry, Pharmacology +5