Concepedia

Evaluation of ligand selectivity using reporter cell lines stably expressing estrogen receptor alpha or beta

Aurélie Escande, Arnaud Pillon, Nadège Servant, Jean‐Pierre Cravedi, Fernando Larrea, Peter Muhn, Jean‐Claude Nicolas, Vincent Cavaillès, Patrick Balaguer

Biochemical Pharmacology · 2006 · 202 citations · 28 references

DOI

Concepts

References

28

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.9K citations

, , +14

Comparison of the Ligand Binding Specificity and Transcript Tissue Distribution of Estrogen Receptors α and β

George G. J. M. Kuiper, Bo Carlsson, Kaj Grandien et al. · Endocrinology · 1997 · 4.4K citations · Full text

, , +14

Interaction of Estrogenic Chemicals and Phytoestrogens with Estrogen Receptor β

George G. J. M. Kuiper, Josephine G. Lemmen, Bo Carlsson et al. · Endocrinology · 1998 · 4.2K citations

, , +17

Molecular basis of agonism and antagonism in the oestrogen receptor

A.M. Brzozowski, A.C.W. Pike, Zbigniew Dauter et al. · Nature · 1997 · 3.3K citations

, , +14

ERβ: Identification and characterization of a novel human estrogen receptor

Sietse Mosselman, Jan Polman, R. Dijkema · FEBS Letters · 1996 · 2.3K citations · Full text

, , +15