Concepedia

Binding characteristics of DAA1106, a novel and selective ligand for peripheral benzodiazepine receptors

Shigeyuki Chaki, Takeo Funakoshi, Ryoko Yoshikawa, Shigeru Okuyama, Taketoshi Okubo, Atsuro Nakazato, Masashi Nagamine, Kazuyuki Tomisawa

European Journal of Pharmacology · 1999 · 80 citations · 24 references

DOI

Concepts

References

24

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.9K citations

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REGIONAL STUDIES OF CATECHOLAMINES IN THE RAT BRAIN‐I

Jacques Glowinski, Leslie L. Iversen · Journal of Neurochemistry · 1966 · 5.4K citations

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Benzodiazepine Receptor: Demonstration in the Central Nervous System

H Möhler, Toshikazu Okada · Science · 1977 · 1.7K citations

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Specific benzodiazepine receptors in rat brain characterized by high-affinity (3H)diazepam binding.

Richard F. Squires · Proceedings of the National Academy of Sciences · 1977 · 1.3K citations · Full text

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GABAergic modulation of benzodiazepine binding site sensitivity

John F. Tallman, John W. Thomas, Dorothy W. Gallager · Nature · 1978 · 725 citations

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