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Novel dual inhibitors of calpain and lipid peroxidation with enhanced cellular activity

Bernadette Pignol, Edith Navet, Morgane Troadec, Denis Carré, José Camara, Dennis Bigg, Pierre‐E. Chabrier

Bioorganic & Medicinal Chemistry Letters · 2005 · 10 citations · 15 references

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15

Novel Peptidyl α-Keto Amide Inhibitors of Calpains and Other Cysteine Proteases

Zhaozhao Li, Anne-Cécile Ortega-Vilain, Girish S. Patil et al. · Journal of Medicinal Chemistry · 1996 · 157 citations · Full text

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Phenothiazine Inhibitors of Trypanothione Reductase as Potential Antitrypanosomal and Antileishmanial Drugs

Cecil Chan, Hong Yin, Jacqui Garforth et al. · Journal of Medicinal Chemistry · 1998 · 140 citations · Full text

, , +15

Peptide .alpha.-keto ester, .alpha.-keto amide, and .alpha.-keto acid inhibitors of calpains and other cysteine proteases

Zhaozhao Li, Girish S. Patil, Zbigniew E. Golubski et al. · Journal of Medicinal Chemistry · 1993 · 109 citations · Full text

, , +14

1,2-Benzothiazine 1,1-dioxide α-ketoamide analogues as potent calpain I inhibitors

Ron Bihovsky, Ming Tao, John P. Mallamo et al. · Bioorganic & Medicinal Chemistry Letters · 2004 · 78 citations · Full text

, , +8

Benzoylalanine-Derived Ketoamides Carrying Vinylbenzyl Amino Residues:  Discovery of Potent Water-Soluble Calpain Inhibitors with Oral Bioavailability

W. Lubisch, Edith Beckenbach, Sabina Bopp et al. · Journal of Medicinal Chemistry · 2003 · 67 citations · Full text

, , +13