W. Lubisch

Discovery and SAR of 2-(1-propylpiperidin-4-yl)-1H-benzimidazole-4-carboxamide: A potent inhibitor of poly(ADP-ribose) polymerase (PARP) for the treatment of cancer

Thomas D. Penning, Gui‐Dong Zhu, Viraj B. Gandhi et al. · Bioorganic & Medicinal Chemistry · 2008 · 75 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +9

Benzoylalanine-Derived Ketoamides Carrying Vinylbenzyl Amino Residues:  Discovery of Potent Water-Soluble Calpain Inhibitors with Oral Bioavailability

W. Lubisch, Edith Beckenbach, Sabina Bopp et al. · Journal of Medicinal Chemistry · 2003 · 67 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +13

A new pyrrolyl‐quinoxalinedione series of non‐NMDA glutamate receptor antagonists: pharmacological characterization and comparison with NBQX and valproate in the kindling model of epilepsy

Wolfgang Löscher, Holger Lehmann, Berthold Behl et al. · European Journal of Neuroscience · 1999 · 52 citations

Medicine, Medicinal Chemistry, Pharmacology +16

Potent and selective oxindole-based vasopressin 1b receptor antagonists with improved pharmacokinetic properties

Thorsten Oost, Gisela Backfisch, Swati Bhowmik et al. · Bioorganic & Medicinal Chemistry Letters · 2011 · 46 citations · Full text

Medicine, Pharmacokinetics, Pharmacology +8

Synthesis and biological evaluation of novel piperidine carboxamide derived calpain inhibitors

W. Lubisch, H. P. Hofmann, Hannes Treiber et al. · Bioorganic & Medicinal Chemistry Letters · 2000 · 28 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +15