Concepedia

Boro-norleucine as a P1 residue for the design of selective and potent DPP7 inhibitors

Kevin Shreder, Melissa S. Wong, Sergio Corral, Zhizhou Yu, David T. Winn, Min Wu, Yi Hu, Tyzoon Nomanbhoy, Senaiet Alemayehu, Stacy R. Fuller,

Bioorganic & Medicinal Chemistry Letters · 2005 · 15 citations · 21 references

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21

Dipeptidyl‐peptidase IV hydrolyses gastric inhibitory polypeptide, glucagon‐like peptide‐1(7–36)amide, peptide histidine methionine and is responsible for their degradation in human serum

Rolf Mentlein, Baptist Gallwitz, Wolfgang E. Schmidt · European Journal of Biochemistry · 1993 · 1.2K citations · Full text

, , +17

Discovering potent and selective reversible inhibitors of enzymes in complex proteomes

Donmienne Leung, Christophe Hardouin, Dale L. Boger et al. · Nature Biotechnology · 2003 · 385 citations

, , +11

Catalytic properties and inhibition of proline-specific dipeptidyl peptidases II, IV and VII

Barbara Leiting, KellyAnn D. Pryor, Joseph K. Wu et al. · Biochemical Journal · 2003 · 181 citations · Full text

, , +15

Structure−Activity Relationships of Boronic Acid Inhibitors of Dipeptidyl Peptidase IV. 1. Variation of the P<sub>2</sub>Position of X<sub>aa</sub>-boroPro Dipeptides

Simon J. Coutts, Terence A. Kelly, Roger J. Snow et al. · Journal of Medicinal Chemistry · 1996 · 123 citations · Full text

, , +17

Two efficient methods for the cleavage of pinanediol boronate esters yielding the free boronic acids

Simon J. Coutts, Julian Adams, Dale A. Krolikowski et al. · Tetrahedron Letters · 1994 · 106 citations

, , +8