Simon J. Coutts

Structure−Activity Relationships of Boronic Acid Inhibitors of Dipeptidyl Peptidase IV. 1. Variation of the P₂Position of X_aa-boroPro Dipeptides

Simon J. Coutts, Terence A. Kelly, Roger J. Snow et al. · Journal of Medicinal Chemistry · 1996 · 122 citations · Full text

Bioorganic Chemistry, Cell Culture, Peptide Science +19

Two efficient methods for the cleavage of pinanediol boronate esters yielding the free boronic acids

Simon J. Coutts, Julian Adams, Dale A. Krolikowski et al. · Tetrahedron Letters · 1994 · 105 citations

Engineering, Pinanediol Boronate Esters, Free Boronic Acids +8

Effect of Structural Modification of Enol−Carboxamide-Type Nonsteroidal Antiinflammatory Drugs on COX-2/COX-1 Selectivity

Edward S. Lazer, Clara K. Miao, Charles L. Cywin et al. · Journal of Medicinal Chemistry · 1997 · 92 citations · Full text

Studies on Proline Boronic Acid Dipeptide Inhibitors of Dipeptidyl Peptidase IV: Identification of a Cyclic Species Containing a B-N Bond

Roger J. Snow, William W. Bachovchin, Randall W. Barton et al. · Journal of the American Chemical Society · 1994 · 78 citations

Pharmaceutical Science, Bioorganic Chemistry, Altmetric Attention Score +21

Immunosuppresive boronic acid dipeptides: correlation between conformation and activity

Terence A. Kelly, Julian Adams, William W. Bachovchin et al. · Journal of the American Chemical Society · 1993 · 42 citations

Medicinal Chemistry, Molecular Sciences, Pharmaceutical Science +15