Nature Chemistry · 2015 · 219 citations · 32 references
PharmacyMedicinal ChemistryDrug DesignDrug DiscoveryMolecular RecognitionLigand BindingLigand-based DesignProtein-ligand BindingProtein-ligand InteractionsProtein-ligand RecognitionReceptor-ligand InteractionsAffinity OptimizationAntibody Affinity MaturationBinding Affinity EnhancementLigand PreparationLigand-receptor AffinityTarget-ligand Interactions
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In vitro selection of RNA molecules that bind specific ligands
Andrew D. Ellington, Jack W. Szostak · Nature · 1990 · 9.7K citations
Phage antibodies: filamentous phage displaying antibody variable domains
John McCafferty, Andrew D. Griffiths, Greg Winter et al. · Nature · 1990 · 2.4K citations
Discovering High-Affinity Ligands for Proteins: SAR by NMR
Suzanne B. Shuker, Philip J. Hajduk, Robert Meadows et al. · Science · 1996 · 2K citations