Concepedia
Naunyn-Schmiedeberg s Archives of Pharmacology · 2008 · 58 citations · 61 references
Signal TransductionFunctional SelectivityMedicinePhysiologyMechanism Of ActionReceptor (Biochemistry)Vitro Pharmacological ProfileExperimental PharmacologyPharmacotherapyHigh Intrinsic ActivityPharmacologyDrug Discovery
61
Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction
Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.8K citations
Cent Inhibition, Inhibitory Activity, Biochemistry +8
A highly sensitive adenylate cyclase assay
Yoram Salomon, Constantine Londos, Martin Rodbell · Analytical Biochemistry · 1974 · 4.2K citations
Cellular Enzymology, Biochemistry, Molecular Biological Method +4
Pharmacologic Analysis of Drug Receptor Interaction
Kenakin. T. Kenakin · Therapeutic Drug Monitoring · 1988 · 929 citations
Data Affinity, Drug Interactions, Drug Receptor Interaction +11
Tegaserod, a 5‐HT<sub>4</sub> receptor partial agonist, relieves symptoms in irritable bowel syndrome patients with abdominal pain, bloating and constipation
S. Müller‐Lissner, I. Fumagalli, Karna Dev Bardhan et al. · Alimentary Pharmacology & Therapeutics · 2001 · 464 citations · Full text
Tegaserod accelerates orocecal transit in patients with constipation-predominant irritable bowel syndrome
Charlene M. Prather, Michael Camilleri, Alan R. Zinsmeister et al. · Gastroenterology · 2000 · 412 citations
Functional Gastrointestinal Disorder, Gastroenterology, Orocecal Transit +4