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Pharmacologic Analysis of Drug Receptor Interaction
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1988
Year
Data AffinityDrug InteractionsDrug Receptor InteractionDrug TargetReceptor Classification KineticsBiochemistryDrug Receptor/theory SevenMedicineFunctional SelectivityPharmacotherapySystems BiologyPharmacologyDrug DiscoveryDrug Resistance
Drug receptor/theory seven transmembrane receptor behaviour human recombinant receptor systems stimulus-response mechanisms drug response mechanisms diffusion and drug concentration in receptor compartments statistical assessment of biological significance from data affinity efficacy competitive antagonism allotopic, noncompetitive, and irreversible antagonism methods of drug and receptor classification kinetics of drug and reaction.