Hybrid diarylbenzopyrimidine non-nucleoside reverse transcriptase inhibitors as promising new leads for improved anti-HIV-1 chemotherapy

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Rapid and automated tetrazolium-based colorimetric assay for the detection of anti-HIV compounds

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Medicinal Chemistry, Bioassay-guided Isolation, Tetrazolium-based Colorimetric Assay +12

Roles of Conformational and Positional Adaptability in Structure-Based Design of TMC125-R165335 (Etravirine) and Related Non-nucleoside Reverse Transcriptase Inhibitors That Are Highly Potent and Effective against Wild-Type and Drug-Resistant HIV-1 Variants

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Tetrazolium-based colorimetric assay for the detection of HIV replication inhibitors: revisited 20 years later

Christophe Pannecouque, Dirk Daelemans, Erik De Clercq · Nature Protocols · 2008 · 347 citations

Hiv Replication Inhibitors, Medicinal Chemistry, Medicine +13

Evolution of Anti-HIV Drug CandidatesPart 2: Diaryltriazine (DATA) Analogues

Donald Ludovici, Robert W. Kavash, Michael J. Kukla et al. · Bioorganic & Medicinal Chemistry Letters · 2001 · 125 citations

Medicinal Chemistry, Medicine, Antiviral Drug Development +7