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1,2-disubstituted indole, azaindole and benzimidazole derivatives possessing amine moiety: a novel series of thrombin inhibitors

DOI

35

Citations

4

References

2000

Year

Kumiko Takeuchi, Jolie Bastian, Donetta S. Gifford‐Moore, Richard W. Harper, Shawn C. Miller, Jeffrey T. Mullaney, Daniel J. Sall, Gerald F. Smith, Minsheng Zhang, Matthew J. Fisher
Bioorganic & Medicinal Chemistry Letters

References

YearCitations

Dibasic Benzo[<i>b</i>]thiophene Derivatives as a Novel Class of Active Site-Directed Thrombin Inhibitors. 1. Determination of the Serine Protease Selectivity, Structure−Activity Relationships, and Binding Orientation

Daniel J. Sall, Jolie Bastian, John A. Buben,

Journal of Medicinal Chemistry

1997

54

Dibasic benzo[b]thiophene derivatives as a novel class of active site directed thrombin inhibitors: 4. SAR studies on the conformationally restricted C3-side chain of hydroxybenzo[b]thiophenes

Kumiko Takeuchi, Todd J. Kohn, Daniel J. Sall,

Bioorganic & Medicinal Chemistry Letters

1999

35

Diamino Benzo[<i>b</i>]thiophene Derivatives as a Novel Class of Active Site Directed Thrombin Inhibitors. 5. Potency, Efficacy, and Pharmacokinetic Properties of Modified C-3 Side Chain Derivatives

Daniel J. Sall, Dianna L. Bailey, Jolie Bastian,

Journal of Medicinal Chemistry

2000

30

Dibasic benzo[b]thiophene derivatives as a novel class of active site directed thrombin inhibitors: 2: sidechain optimization and demonstration of in vivo efficacy

Minsheng Zhang, Dianna L. Bailey, Jolie Bastian,

Bioorganic & Medicinal Chemistry Letters

1999

13

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