Potent and selective inhibitors of PI3Kδ: Obtaining isoform selectivity from the affinity pocket and tryptophan shelf - Concepedia

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Potent and selective inhibitors of PI3Kδ: Obtaining isoform selectivity from the affinity pocket and tryptophan shelf

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50

Citations

15

References

2012

Year

Daniel P. Sutherlin, Stewart Baker, Angelina Bisconte, Paul Blaney, Anthony Brown, Bryan Chan, David Chantry, Georgette M. Castanedo, Paul Depledge, Paul Goldsmith,

Bioorganic & Medicinal Chemistry Letters

BiochemistryFunctional SelectivityMedicinePharmacologyRational Drug DesignAffinity PocketIsoform SelectivityMolecular DockingTryptophan ShelfInhibitory ActivityDrug Discovery

References

	Year	Citations

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