Concepedia

Characterization of Non-peptide Antagonist and Peptide Agonist Binding Sites of the NK1 Receptor with Fluorescent Ligands

Gerardo Turcatti, Sannah Zoffmann, John Lowe, Susan E. Drozda, Gérard Chassaing, Thue W. Schwartz, André Chollet

Journal of Biological Chemistry · 1997 · 62 citations · 34 references

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References

34

A Potent Nonpeptide Antagonist of the Substance P (NK <sub>1</sub> ) Receptor

R. Michael Snider, Jay W. Constantine, John Lowe et al. · Science · 1991 · 864 citations

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Discovery of a potent substance P antagonist: recognition of the key molecular determinant

Manoj C. Desai, Sheri L. Lefkowitz, Peter F. Thadeio et al. · Journal of Medicinal Chemistry · 1992 · 220 citations · Full text

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Different binding epitopes on the NK1 receptor for substance P and a non-peptide antagonist

Ulrik Gether, Teit E. Johansen, R. Michael Snider et al. · Nature · 1993 · 218 citations

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Activity and Distribution of Binding Sites in Brain of a Nonpeptide Substance P (NK <sub>1</sub> ) Receptor Antagonist

Stafford McLean, Alan H. Ganong, Thomas Seeger et al. · Science · 1991 · 218 citations

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Localization of agonist and antagonist binding domains of the human neurokinin-1 receptor.

Tung M. Fong, R R Huang, Catherine D. Strader · Journal of Biological Chemistry · 1992 · 193 citations · Full text

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